DrugDomain logoDrugDomain

N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide

P10721 — Mast/stem cell growth factor receptor Kit

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Attributes

UniProt ID
P10721
Protein Name
Mast/stem cell growth factor receptor Kit
Ligand Name
N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide
DrugBank ID
DB01268
PDB Ligand Accession
B49
ChEMBL ID
CHEMBL535
PubChem ID
5329102
InChIKey
WINHZLLDWRZWRT-ATVHPVEESA-N
SMILES
CCN(CC)CCNC(=O)c1c(c([nH]c1C)C=C2c3cc(ccc3NC2=O)F)C
Drug Action
inhibitor
Affinity Metrics
ki:4 nM
ic50:0.8 nM
kd:0.21 nM