Pirenzepine

P11229 — Muscarinic acetylcholine receptor M1

Attributes

UniProt ID

Protein Name

Muscarinic acetylcholine receptor M1

Ligand Name

Pirenzepine

DrugBank ID

PDB Ligand Accession

n/a

ChEMBL ID

n/a

PubChem ID

n/a

InChIKey

n/a

SMILES

CN1CCN(CC(=O)N2C3=CC=CC=C3C(=O)NC3=C2N=CC=C3)CC1

Drug Action

antagonist

Affinity Metrics

ki:2.82 nM

ic50:1.5 nM

kd:20 nM