DrugDomain logoDrugDomain

5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide

P21554 — Cannabinoid receptor 1

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Attributes

UniProt ID
P21554
Protein Name
Cannabinoid receptor 1
Ligand Name
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
DrugBank ID
DB06155
PDB Ligand Accession
AY6
ChEMBL ID
CHEMBL111
PubChem ID
104850
InChIKey
JZCPYUJPEARBJL-UHFFFAOYSA-N
SMILES
Cc1c(n(nc1C(=O)NN2CCCCC2)c3ccc(cc3Cl)Cl)c4ccc(cc4)Cl
Drug Action
antagonist
Affinity Metrics
ki:0.4 nM
ic50:1.35 nM
kd:1.8 nM
ec50:0.11 nM