Sitaxentan

P25101 — Endothelin-1 receptor

Attributes

UniProt ID

Protein Name

Endothelin-1 receptor

Ligand Name

Sitaxentan

DrugBank ID

PDB Ligand Accession

n/a

ChEMBL ID

n/a

PubChem ID

n/a

InChIKey

n/a

SMILES

CC1=NOC(NS(=O)(=O)C2=C(SC=C2)C(=O)CC2=CC3=C(OCO3)C=C2C)=C1Cl

Drug Action

antagonist

Affinity Metrics

ki:0.43 nM

ic50:1.4 nM