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N,N-diethyl-N'-[(8alpha)-6-methyl-9,10-didehydroergolin-8-yl]urea

P28223 — 5-hydroxytryptamine receptor 2A

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Attributes

UniProt ID
P28223
Protein Name
5-hydroxytryptamine receptor 2A
Ligand Name
N,N-diethyl-N'-[(8alpha)-6-methyl-9,10-didehydroergolin-8-yl]urea
DrugBank ID
DB00589
PDB Ligand Accession
H8G
ChEMBL ID
CHEMBL157138
PubChem ID
28864
InChIKey
BKRGVLQUQGGVSM-KBXCAEBGSA-N
SMILES
CCN(CC)C(=O)NC1CN(C2Cc3c[nH]c4c3c(ccc4)C2=C1)C
Drug Action
agonist
Affinity Metrics
ki:5.4 nM
ic50:0.97 nM
ec50:343 nM