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4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol

P29274 — Adenosine receptor A2a

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Attributes

UniProt ID
P29274
Protein Name
Adenosine receptor A2a
Ligand Name
4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol
DrugBank ID
DB08770
PDB Ligand Accession
ZMA
ChEMBL ID
CHEMBL113142
PubChem ID
176407
InChIKey
PWTBZOIUWZOPFT-UHFFFAOYSA-N
SMILES
c1cc(oc1)c2nc3nc(nc(n3n2)N)NCCc4ccc(cc4)O
Drug Action
inhibitor
Affinity Metrics
ki:0.1 nM
ic50:0.678 nM
kd:0.22 nM