Tiagabine
P30531 — Sodium- and chloride-dependent GABA transporter 1
Attributes
UniProt ID
Protein Name
Sodium- and chloride-dependent GABA transporter 1
Ligand Name
Tiagabine
DrugBank ID
PDB Ligand Accession
ChEMBL ID
InChIKey
PBJUNZJWGZTSKL-MRXNPFEDSA-N
SMILES
Cc1ccsc1C(=CCCN2CCCC(C2)C(=O)O)c3c(ccs3)C
Drug Action
inhibitor
Affinity Metrics
ki:16.98 nM
ic50:49 nM
kd:41 nM