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2,4-THIAZOLIDIINEDIONE, 5-[[4-[2-(METHYL-2-PYRIDINYLAMINO)ETHOXY]PHENYL]METHYL]-(9CL)

P37231 — Peroxisome proliferator-activated receptor gamma

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Attributes

UniProt ID
P37231
Protein Name
Peroxisome proliferator-activated receptor gamma
Ligand Name
2,4-THIAZOLIDIINEDIONE, 5-[[4-[2-(METHYL-2-PYRIDINYLAMINO)ETHOXY]PHENYL]METHYL]-(9CL)
DrugBank ID
DB00412
PDB Ligand Accession
BRL
ChEMBL ID
CHEMBL121106
PubChem ID
445655
InChIKey
YASAKCUCGLMORW-HNNXBMFYSA-N
SMILES
CN(CCOc1ccc(cc1)CC2C(=O)NC(=O)S2)c3ccccn3
Drug Action
agonist
Affinity Metrics
ki:8 nM
ic50:7.7 nM
kd:1.2 nM
ec50:1 nM
koff:0.145 nM