DrugDomain logoDrugDomain

4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimidazol-3'-yl)methyl]biphenyl-2-carboxylic acid

P37231 — Peroxisome proliferator-activated receptor gamma

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Attributes

UniProt ID
P37231
Protein Name
Peroxisome proliferator-activated receptor gamma
Ligand Name
4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimidazol-3'-yl)methyl]biphenyl-2-carboxylic acid
DrugBank ID
DB00966
PDB Ligand Accession
TLS
ChEMBL ID
CHEMBL1017
PubChem ID
65999
InChIKey
RMMXLENWKUUMAY-UHFFFAOYSA-N
SMILES
CCCc1nc2c(cc(cc2n1Cc3ccc(cc3)c4ccccc4C(=O)O)c5nc6ccccc6n5C)C
Drug Action
partial agonist
Affinity Metrics
ki:1080 nM
ic50:12200 nM
ec50:700 nM