DrugDomain logoDrugDomain

VARENICLINE

P43681 — Neuronal acetylcholine receptor subunit alpha-4

← Back

Attributes

UniProt ID
P43681
Protein Name
Neuronal acetylcholine receptor subunit alpha-4
Ligand Name
VARENICLINE
DrugBank ID
DB01273
PDB Ligand Accession
QMR
ChEMBL ID
CHEMBL1076903
PubChem ID
5310966
InChIKey
JQSHBVHOMNKWFT-DTORHVGOSA-N
SMILES
c1cnc2cc3c(cc2n1)C4CC3CNC4
Drug Action
partial agonist
Affinity Metrics
ki:0.04 nM
ic50:94 nM
ec50:950 nM