DB00543
Proteins interacting with this molecule.
| DrugDomain Data | DrugBank | PDB Ligand | UniProt | Protein Name | Drug Action | Affinity |
|---|---|---|---|---|---|---|
| Explore | DB00543 | n/a | P08908 | 5-hydroxytryptamine receptor 1A | antagonist | Ki 221 nM |
| Explore | DB00543 | n/a | P08913 | Alpha-2A adrenergic receptor | antagonist | n/a |
| Explore | DB00543 | n/a | P11229 | Muscarinic acetylcholine receptor M1 | antagonist | n/a |
| Explore | DB00543 | n/a | P14416 | D dopamine receptor | antagonist | Ki 3.6 nM |
| Explore | DB00543 | n/a | P14867 | Gamma-aminobutyric acid receptor subunit alpha-1 receptor subunit alpha-1 | binder | n/a |
| Explore | DB00543 | n/a | P21728 | D dopamine receptor | antagonist | n/a |
| Explore | DB00543 | n/a | P21917 | D dopamine receptor dopamine receptor | antagonist | Ki 2 nM |
| Explore | DB00543 | n/a | P23975 | Sodium-dependent noradrenaline transporter | inhibitor | Ki 16 nM |
| Explore | DB00543 | n/a | P28222 | 5-hydroxytryptamine receptor 1B | antagonist | n/a |
| Explore | DB00543 | n/a | P28223 | 5-hydroxytryptamine receptor 2A | antagonist | Ki 1.77 nM |
| Explore | DB00543 | n/a | P28335 | 5-hydroxytryptamine receptor 2C | antagonist | n/a |
| Explore | DB00543 | n/a | P31645 | Sodium-dependent serotonin transporter | inhibitor | Ki 58 nM |
| Explore | DB00543 | n/a | P34969 | 5-hydroxytryptamine receptor 7 | antagonist | Ki 500 nM |
| Explore | DB00543 | n/a | P35348 | Alpha-1A adrenergic receptor | antagonist | n/a |
| Explore | DB00543 | n/a | P35367 | Histamine H1 receptor | antagonist | n/a |
| Explore | DB00543 | n/a | P35462 | D dopamine receptor | antagonist | Ki 11 nM |
| Explore | DB00543 | n/a | P41595 | 5-hydroxytryptamine receptor 2B | antagonist | n/a |
| Explore | DB00543 | n/a | P46098 | 5-hydroxytryptamine receptor 3A | antagonist | n/a |
| Explore | DB00543 | n/a | P50406 | 5-hydroxytryptamine receptor 6 | antagonist | Ki 50 nM |
| Explore | DB00543 | n/a | Q01959 | Sodium-dependent dopamine transporter | binder | Ki 4310 nM |
Showing 20 of 21 interactions