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0LI

Proteins interacting with this PDB ligand.

DrugDomain DataDrugBank IDPDB LigandUniProtProtein NameDrug ActionAffinity
ExploreDB089010LID3DSX2deletedno_target_actionn/a
ExploreDB089010LIO43353Receptor-interacting serine/threonine-protein kinase 2no_target_actionIC50 1 nM
ExploreDB089010LIP00519Tyrosine-protein kinase ABL1inhibitorIC50 0.3 nM | Kd 0.7 nM | EC50 0.05 nM
ExploreDB089010LIP00520Tyrosine-protein kinase ABL1no_target_actionn/a
ExploreDB089010LIP00523Proto-oncogene tyrosine-protein kinase Srcno_target_actionIC50 0.9 nM | Kd 0.7 nM
ExploreDB089010LIP06239Tyrosine-protein kinase LckinhibitorIC50 0.28 nM
ExploreDB089010LIP07948Tyrosine-protein kinase LyninhibitorIC50 0.16 nM
ExploreDB089010LIP07949Proto-oncogene tyrosine-protein kinase receptor RetinhibitorIC50 0.3 nM
ExploreDB089010LIP10721Mast/stem cell growth factor receptor KitinhibitorIC50 1.7 nM
ExploreDB089010LIP11274Breakpoint cluster region proteininhibitorn/a
ExploreDB089010LIP11362Fibroblast growth factor receptor 1inhibitorIC50 0.7 nM
ExploreDB089010LIP12931Proto-oncogene tyrosine-protein kinase SrcinhibitorIC50 2.5 nM
ExploreDB089010LIP15056Serine/threonine-protein kinase B-rafno_target_actionn/a
ExploreDB089010LIP16234Platelet-derived growth factor receptor alphainhibitorIC50 1.1 nM
ExploreDB089010LIP21802Fibroblast growth factor receptor 2inhibitorIC50 1.3 nM
ExploreDB089010LIP22455Fibroblast growth factor receptor 4inhibitorIC50 7.1 nM
ExploreDB089010LIP22607Fibroblast growth factor receptor 3inhibitorIC50 9.4 nM
ExploreDB089010LIP35968Vascular endothelial growth factor receptor 2inhibitorKi 1.5 nM | IC50 1.5 nM
ExploreDB089010LIP36888Receptor-type tyrosine-protein kinase FLT3inhibitorIC50 0.3 nM
ExploreDB089010LIQ01973Inactive tyrosine-protein kinase transmembrane receptor ROR1no_target_actionn/a
ExploreDB089010LIQ02763Angiopoietin-1 receptorinhibitorn/a
ExploreDB089010LIQ08345Epithelial discoidin domain-containing receptor 1no_target_actionIC50 9.4 nM
ExploreDB089010LIQ9NWZ3Interleukin-1 receptor-associated kinase 4no_target_actionn/a