Gene name: PLK4
Protein name: Serine/threonine-protein kinase PLK4
List of molecules and drugs that interact with protein O00444
# | DrugDomain Data | PBD ligand | DrugBank Accession | PubChem | ChEMBL | Name | Drug action | Affinity data |
---|---|---|---|---|---|---|---|---|
1 | O00444_4J7 | 4J7 | n/a | 91801159 | CHEMBL5185225 | 2-({2-fluoro-4-[(2-fluoro-3-nitrobenzyl)sulfonyl]phenyl}sulfanyl)-5-methoxy-N-(3-methyl-1H-pyrazol-5-yl)-6-(morpholin-4-yl)pyrimidin-4-amine | n/a | |
2 | O00444_631 | 631 | n/a | 58486384 | CHEMBL3353348 | (1R,2S)-2-{3-[(E)-2-{4-[(dimethylamino)methyl]phenyl}ethenyl]-2H-indazol-6-yl}-5'-methoxyspiro[cyclopropane-1,3'-indol]-2'(1'H)-one | n/a | |
3 | O00444_ANP | ANP | n/a | 33113 | CHEMBL1230989 | PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER | n/a | |
4 | O00444_CL | CL | n/a | 312 | n/a | CHLORIDE ION | n/a | |
5 | O00444_SO4 | SO4 | DB14546 | 1117 | n/a | SULFATE ION | n/a | |
6 | O00444_2RC | 2RC | DB12010 | 11671467 | CHEMBL2103830 | Fostamatinib | inhibitor |