P43220 GLP1R_HUMAN
Gene name: GLP1R
Protein name: Glucagon-like peptide 1

List of molecules and drugs that interact with protein P43220

# DrugDomain Data PBD ligand DrugBank Accession PubChem ChEMBL Name Drug action Affinity data
1 P43220_10M 10M n/a 10345813 n/a decyl 4-O-alpha-D-glucopyranosyl-1-thio-beta-D-glucopyranoside n/a
2 P43220_32M 32M n/a 12398655 n/a 3,6,9,12,15,18-hexaoxahexacosan-1-ol n/a
3 P43220_82L 82L n/a 134611223 CHEMBL5191519 2-[(4-{6-[(2,4-difluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-benzimidazole-6-carboxylic acid n/a
4 P43220_97V 97V n/a 23549991 CHEMBL4758265 4-{[(4-cyclohexylphenyl){[3-(methylsulfonyl)phenyl]carbamoyl}amino]methyl}-N-(1H-tetrazol-5-yl)benzamide n/a
5 P43220_97Y 97Y n/a 68178630 CHEMBL3648185 N-{4-[(R)-(3,3-dimethylcyclobutyl)({6-[4-(trifluoromethyl)-1H-imidazol-1-yl]pyridin-3-yl}amino)methyl]benzene-1-carbonyl}-beta-alanine n/a
6 P43220_BYI BYI n/a n/a CHEMBL2158411 2,4-bis(3-methoxy-4-thiophen-2-ylcarbonyloxy-phenyl)-1,3-bis[[4-[(2-methylpropan-2-yl)oxycarbonylamino]phenyl]carbonylamino]cyclobutane-1,3-dicarboxylic acid n/a
7 P43220_CLR CLR DB04540 5997 CHEMBL112570 CHOLESTEROL n/a
8 P43220_D6M D6M n/a 161955 n/a N-hexadecanoyl-L-glutamic acid n/a
9 P43220_FFR FFR n/a 149050799 n/a 2-[[4-[6-[(4-cyano-2-fluoranyl-phenyl)methoxy]pyridin-2-yl]-3,6-dihydro-2~{H}-pyridin-1-yl]methyl]-3-[[(2~{S})-oxetan-2-yl]methyl]imidazo[4,5-b]pyridine-5-carboxylic acid n/a
10 P43220_HEZ HEZ DB02210 12374 CHEMBL458616 HEXANE-1,6-DIOL n/a
11 P43220_HNO HNO n/a 156022738 n/a N-tert-butyl-6,7-bis(chloranyl)quinoxalin-2-amine n/a
12 P43220_N2V N2V n/a 58327143 CHEMBL3950796 N-{(3S,8S)-3-{4-[(3,4-dichlorophenyl)methoxy]phenyl}-7-[(1S)-1-phenylpropyl]-2,3,6,7,8,9-hexahydro[1,4]dioxino[2,3-g]isoquinoline-8-carbonyl}-4-(2,3-dimethylpyridin-4-yl)-L-phenylalanine n/a
13 P43220_NAG NAG DB00141 24139 CHEMBL447878 2-acetamido-2-deoxy-beta-D-glucopyranose n/a
14 P43220_OLA OLA n/a 445639 CHEMBL8659 OLEIC ACID n/a
15 P43220_OLC OLC n/a 11451146 n/a (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate n/a
16 P43220_QW7 QW7 n/a 146155955 CHEMBL5197819 1-[(1R)-1-(2,6-dichloro-3-methoxyphenyl)ethyl]-6-{2-[(2R)-piperidin-2-yl]phenyl}-1H-benzimidazole n/a
17 P43220_SO4 SO4 DB14546 1117 n/a SULFATE ION n/a
18 P43220_UK1 UK1 n/a 154584718 n/a 3-{(1S)-1-[5-(2,2-dimethylmorpholin-4-yl)-2-{(4S)-2-(4-fluoro-3,5-dimethylphenyl)-3-[3-(4-fluoro-1-methyl-1H-indazol-5-yl)-2-oxo-2,3-dihydro-1H-imidazol-1-yl]-4-methyl-2,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indol-1-yl]butyl}-1,2,4-oxadiazol-5(4H)-one n/a
19 P43220_UK4 UK4 DB16043 134611040 CHEMBL4518483 2-[(4-{6-[(4-cyano-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-benzimidazole-6-carboxylic acid agonist
20 P43220_V6G V6G DB18964 137319706 CHEMBL4446782 3-[(1S,2S)-1-(5-[(4S)-2,2-dimethyloxan-4-yl]-2-{(4S)-2-(4-fluoro-3,5-dimethylphenyl)-3-[3-(4-fluoro-1-methyl-1H-indazol-5-yl)-2-oxo-2,3-dihydro-1H-imidazol-1-yl]-4-methyl-2,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indol-1-yl)-2-methylcyclopropyl]-1,2,4-oxadiazol-5(4H)-one agonist
21 P43220_WB2 WB2 n/a n/a CHEMBL2158488 2,4-bis(3-methoxy-4-thiophen-2-ylcarbonyloxy-phenyl)-1,3-bis[[4-(2-methylpropanoylamino)phenyl]carbonylamino]cyclobutane-1,3-dicarboxylic acid n/a
22 P43220_WF1 WF1 n/a 51340918 n/a 17-amino-10-oxo-3,6,12,15-tetraoxa-9-azaheptadecan-1-oic acid n/a
23 P43220_SOG SOG DB08558 656909 n/a octyl 1-thio-beta-D-glucopyranoside n/a
24 P43220_DB13928 n/a DB13928 n/a n/a Semaglutide agonist
25 P43220_DB14027 n/a DB14027 n/a n/a Taspoglutide agonist