1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-3-methyl-6-[6-(piperazin-1-yl)pyridin-3-yl]-1H-indole-4-carboxamide
G0SDW4 — Histone-lysine N-methyltransferase EZH2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand A9G
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand A9G
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| G0SDW4 | n/a | 5wf7 | A9G | B | 8009 | e5wf7B4 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_N |
| G0SDW4 | n/a | 5wf7 | A9G | B | 8009 | e5wf7B8 | beta-clip | SET domain-like | SET domain-like | SET |
| G0SDW4 | n/a | 5wfd | A9G | B | 8009 | e5wfdB4 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_N |
| G0SDW4 | n/a | 5wfd | A9G | B | 8009 | e5wfdB6 | beta-clip | SET domain-like | SET domain-like | SET |