5,8-dichloro-2-[(4-ethyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-7-({1-[(2R)-2-hydroxypropanoyl]piperidin-4-yl}oxy)-3,4-dihydroisoquinolin-1(2H)-one
G1KPH4 — Histone-lysine N-methyltransferase EZH2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 6BN
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 6BN
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| G1KPH4 | n/a | 5ij7 | 6BN | A | 9001 | e5ij7A1 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | n/a | 5ij7 | 6BN | A | 9001 | e5ij7A2 | beta-clip | SET domain-like | SET domain-like | SET |
| G1KPH4 | n/a | 5ij7 | 6BN | B | 9001 | e5ij7B1 | beta-clip | SET domain-like | SET domain-like | SET |
| G1KPH4 | n/a | 5ij7 | 6BN | B | 9001 | e5ij7B2 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | n/a | 5ij8 | 6BN | A | 9001 | e5ij8A1 | beta-clip | SET domain-like | SET domain-like | SET |
| G1KPH4 | n/a | 5ij8 | 6BN | A | 9001 | e5ij8A7 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | n/a | 5ij8 | 6BN | B | 9001 | e5ij8B3 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | n/a | 5ij8 | 6BN | B | 9001 | e5ij8B7 | beta-clip | SET domain-like | SET domain-like | SET |