5,8-dichloro-2-[(4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-7-[(R)-methoxy(oxetan-3-yl)methyl]-3,4-dihydroisoquinolin-1(2H)-one
G1KPH4 — Histone-lysine N-methyltransferase EZH2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand DB14799
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand DB14799
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| G1KPH4 | DB14799 | 4w2r | CJD | A | 708 | e4w2rA5 | beta-clip | SET domain-like | SET domain-like | SET |
| G1KPH4 | DB14799 | 4w2r | CJD | A | 708 | e4w2rA6 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | DB14799 | 4w2r | CJD | B | 708 | e4w2rB6 | Ezh2 N-terminal domain | Ezh2 N-terminal domain | Ezh2 N-terminal domain | EZH2_WD-Binding |
| G1KPH4 | DB14799 | 4w2r | CJD | B | 708 | e4w2rB7 | beta-clip | SET domain-like | SET domain-like | SET |