(2M)-2-[(4M)-4-{4-(aminomethyl)-1-oxo-8-[(2R)-oxolan-2-yl]-1,2-dihydrophthalazin-6-yl}-1-methyl-1H-pyrazol-5-yl]-1-benzothiophene-3-carbonitrile
O14744 — Protein arginine N-methyltransferase 5
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand NXF
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand NXF
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| O14744 | n/a | 7uoh | NXF | A | 801 | e7uohA1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | PRMT5 |
| O14744 | n/a | 7uoh | NXF | A | 801 | e7uohA3 | Arginine methyltransferase oligomerization subdomain | Arginine methyltransferase oligomerization subdomain | Arginine methyltransferase oligomerization subdomain | PRMT5_C |