(7~{R})-2-[[2-ethoxy-4-(1-methylpiperidin-4-yl)phenyl]amino]-7-ethyl-5-methyl-8-(phenylmethyl)-7~{H}-pteridin-6-one
O60885 — Bromodomain-containing protein 4
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand HG5
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand HG5
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| O60885 | n/a | 6q3y | HG5 | A | 202 | e6q3yA1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |
| O60885 | n/a | 6q3y | HG5 | B | 204 | e6q3yA1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |
| O60885 | n/a | 6q3y | HG5 | B | 204 | e6q3yB1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |