3-methyl-6-[6-[(3~{S})-3-methylmorpholin-4-yl]-1-[(1~{S})-1-phenylethyl]imidazo[4,5-c]pyridin-2-yl]-~{N}-propan-2-yl-[1,2,4]triazolo[4,3-a]pyrazin-8-amine
O60885 — Bromodomain-containing protein 4
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand O2B
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand O2B
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| O60885 | n/a | 6xv3 | O2B | A | 4000 | e6xv3A1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |
| O60885 | n/a | 6xv3 | O2B | B | 201 | e6xv3B1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |
| O60885 | n/a | 6xv3 | O2B | C | 201 | e6xv3C1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |
| O60885 | n/a | 6xv3 | O2B | D | 201 | e6xv3D1 | Bromodomain-like | Bromodomain | Bromodomain | Bromodomain |