DrugDomain logoDrugDomain

Attributes

UniProt ID
Protein Name
Isocitrate dehydrogenase cytoplasmic -specific ICDH
Ligand Name
[2-[2-[[1-[4-[(1S)-1-[[5-fluoranyl-4-[(4S)-2-oxidanylidene-4-propan-2-yl-1,3-oxazolidin-3-yl]pyrimidin-2-yl]amino]ethyl]phenyl]piperidin-4-yl]sulfamoyl]ethylsulfanylmethyl]-3-oxidanylidene-propyl]-trimethyl-azanium
DrugBank ID
None
PDB Ligand Accession
ChEMBL ID
n/a
PubChem ID
n/a
InChIKey
LCIIBZXZTLMNNC-QFTSJRPJSA-N
SMILES
CC(C)C1COC(=O)N1c2c(cnc(n2)NC(C)c3ccc(cc3)N4CCC(CC4)NS(=O)(=O)CCSCC(C[N+](C)(C)C)C=O)F
Drug Action
No data available
Affinity Metrics
No affinity data available

3D Structure

Interactive Mol* view for the current protein-molecule pair.

Structure: 8HB9
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Color Legend
Unassigned regionsLigand / hetero atomse8hb9AAA1e8hb9AAA2e8hb9BBB1e8hb9BBB2e8hb9CCC1e8hb9CCC2e8hb9DDD1e8hb9DDD2
ECOD domains from experimental PDB structures interacting with ligand R1R
UniProtDrugBankPDB LigandPDB IDECOD DomainRange Definition
O75874n/aR1R8hb9e8hb9AAA1AAA:106-286
O75874n/aR1R8hb9e8hb9AAA2AAA:3-105,AAA:287-412
O75874n/aR1R8hb9e8hb9BBB1BBB:3-105,BBB:287-412
O75874n/aR1R8hb9e8hb9BBB2BBB:106-286
O75874n/aR1R8hb9e8hb9CCC1CCC:3-105,CCC:287-412
O75874n/aR1R8hb9e8hb9CCC2CCC:106-286
O75874n/aR1R8hb9e8hb9DDD1DDD:1-105,DDD:287-411
O75874n/aR1R8hb9e8hb9DDD2DDD:106-286