3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[4-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]propanamide
O95271 — Poly polymerase tankyrase-1
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 2C8
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 2C8
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| O95271 | n/a | 4msk | 2C8 | A | 1402 | e4mskA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4msk | 2C8 | B | 1402 | e4mskB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4msk | 2C8 | C | 1402 | e4mskC1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4msk | 2C8 | D | 1402 | e4mskD1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |