1-[(1-acetyl-5-bromo-1H-indol-6-yl)sulfonyl]-N-ethyl-N-(3-methylphenyl)piperidine-4-carboxamide
O95271 — Poly polymerase tankyrase-1
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand IW8
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand IW8
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| O95271 | n/a | 4tor | IW8 | A | 1402 | e4torA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4tor | IW8 | B | 1402 | e4torB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4tor | IW8 | C | 1402 | e4torC1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| O95271 | n/a | 4tor | IW8 | D | 1402 | e4torD1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |