(4P)-2-amino-4-{4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-8-fluoro-2-{[(2R,4R,7aS)-2-fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl]methoxy}-6-(trifluoromethyl)quinazolin-7-yl}-7-fluoro-1-benzothiophene-3-carbonitrile
P01116 — GTPase KRas
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand VR5
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand VR5
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| P01116 | n/a | 8txh | VR5 | A | 203 | e8txhA1 | P-loop domains-like | P-loop domains-related | P-loop containing nucleoside triphosphate hydrolases | Ras |
| P01116 | n/a | 8txh | VR5 | B | 203 | e8txhB1 | P-loop domains-like | P-loop domains-related | P-loop containing nucleoside triphosphate hydrolases | Ras |