2-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-thiopyrano[4,3-d]pyrimidin-4-ol
P09874 — Poly polymerase 1 ADP-ribosyltransferase 1) polymerase 1, processed C-terminus ; Poly polymerase 1, processed N-terminus ]
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand XAV
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand XAV
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| P09874 | n/a | 4r5w | XAV | A | 1106 | e4r5wA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| P09874 | n/a | 4r5w | XAV | A | 1106 | e4r5wA2 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | PARP_reg |
| P09874 | n/a | 4r5w | XAV | B | 1103 | e4r5wB1 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | PARP_reg |
| P09874 | n/a | 4r5w | XAV | B | 1103 | e4r5wB2 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |