(4S)-19-acetyl-4-[(1R)-1-hydroxy-2-({1-[3-(propan-2-yl)phenyl]cyclopropyl}amino)ethyl]-11-oxa-3,16-diazatricyclo[15.3.1.1~6,10~]docosa-1(21),6(22),7,9,17,19-hexaen-2-one
P56817 — Beta-secretase 1
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand E4A
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand E4A
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| P56817 | n/a | 5qco | E4A | A | 401 | e5qcoA1 | cradle loop barrel | RIFT-related | acid protease | Asp |
| P56817 | n/a | 5qco | E4A | A | 401 | e5qcoA2 | cradle loop barrel | RIFT-related | acid protease | Asp |
| P56817 | n/a | 5qco | E4A | B | 401 | e5qcoB1 | cradle loop barrel | RIFT-related | acid protease | Asp |
| P56817 | n/a | 5qco | E4A | B | 401 | e5qcoB2 | cradle loop barrel | RIFT-related | acid protease | Asp |
| P56817 | n/a | 5qco | E4A | C | 401 | e5qcoC1 | cradle loop barrel | RIFT-related | acid protease | Asp |
| P56817 | n/a | 5qco | E4A | C | 401 | e5qcoC2 | cradle loop barrel | RIFT-related | acid protease | Asp |