{4-[2-(2-hydroxyethoxy)phenyl]piperazin-1-yl}[(2R,3S)-2-propyl-3-[4-(trifluoromethyl)phenoxy]-1-{[4-(trifluoromethyl)pyridin-3-yl]carbonyl}piperidin-3-yl]methanone
Q00987 — E3 ubiquitin-protein ligase Mdm2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 62Q
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 62Q
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q00987 | n/a | 5hmk | 62Q | A | 1001 | e5hmkA1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 5hmk | 62Q | A | 1001 | e5hmkB1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 5hmk | 62Q | B | 1001 | e5hmkA1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 5hmk | 62Q | B | 1001 | e5hmkB1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |