4-[(4~{S})-5-(5-chloranyl-2-oxidanylidene-1~{H}-pyridin-3-yl)-2-[2-(dimethylamino)-4-methoxy-pyrimidin-5-yl]-6-oxidanylidene-3-propan-2-yl-4~{H}-pyrrolo[3,4-c]pyrazol-4-yl]benzenecarbonitrile
Q00987 — E3 ubiquitin-protein ligase Mdm2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand HRE
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand HRE
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q00987 | n/a | 6q96 | HRE | A | 201 | e6q96A1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q96 | HRE | A | 201 | e6q96B1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q96 | HRE | B | 201 | e6q96A1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q96 | HRE | B | 201 | e6q96B1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |