~{N}-~{tert}-butyl-2-[4-chloranyl-2-[5-(3-chloranyl-4-fluoranyl-phenyl)-2-cyclohexyl-4-(1~{H}-1,2,3,4-tetrazol-5-yl)imidazol-1-yl]phenyl]ethanamide
Q00987 — E3 ubiquitin-protein ligase Mdm2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand HU8
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand HU8
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q00987 | n/a | 6q9o | HU8 | A | 201 | e6q9oA1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q9o | HU8 | A | 201 | e6q9oB1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q9o | HU8 | B | 201 | e6q9oA1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |
| Q00987 | n/a | 6q9o | HU8 | B | 201 | e6q9oB1 | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB/MDM2 domain | SWIB |