DrugDomain logoDrugDomain

Attributes

UniProt ID
Protein Name
Beta-lactamase OXA-48
Ligand Name
(2S,3R,4S)-4-({(3S,5S)-5-[(3-carboxyphenyl)carbamoyl]pyrrolidin-3-yl}sulfanyl)-2-[(1S,2R)-1-formyl-2-hydroxypropyl]-3-methyl-3,4-dihydro-2H-pyrrole-5-carboxylic acid
DrugBank ID
None
PDB Ligand Accession
ChEMBL ID
n/a
PubChem ID
n/a
InChIKey
RALHTEQYPKBGFO-SAGZMZRGSA-N
SMILES
CC1C(C(=NC1C(C=O)C(C)O)C(=O)O)SC2CC(NC2)C(=O)Nc3cccc(c3)C(=O)O
Drug Action
No data available
Affinity Metrics
No affinity data available

3D Structure

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Structure: 6ZRJ
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Color Legend
Unassigned regionsLigand / hetero atomse6zrjA1e6zrjA2e6zrjB1e6zrjB2e6zrjC1e6zrjC2e6zrjD1e6zrjD2e6zrjE1e6zrjE2e6zrjF1e6zrjF2e6zrjG1e6zrjG2e6zrjH1e6zrjH2
ECOD domains from experimental PDB structures interacting with ligand 2RG
UniProtDrugBankPDB LigandPDB IDECOD DomainRange Definition
Q6XEC0n/a2RG6zrje6zrjA1A:23-64,A:162-265
Q6XEC0n/a2RG6zrje6zrjA2A:63-163
Q6XEC0n/a2RG6zrje6zrjB1B:23-64,B:162-265
Q6XEC0n/a2RG6zrje6zrjB2B:63-163
Q6XEC0n/a2RG6zrje6zrjC1C:63-163
Q6XEC0n/a2RG6zrje6zrjC2C:23-64,C:162-265
Q6XEC0n/a2RG6zrje6zrjD1D:24-64,D:162-265
Q6XEC0n/a2RG6zrje6zrjD2D:63-163
Q6XEC0n/a2RG6zrje6zrjE1E:24-64,E:162-265
Q6XEC0n/a2RG6zrje6zrjE2E:63-163
Q6XEC0n/a2RG6zrje6zrjF1F:63-163
Q6XEC0n/a2RG6zrje6zrjF2F:24-64,F:162-265
Q6XEC0n/a2RG6zrje6zrjG1G:63-163
Q6XEC0n/a2RG6zrje6zrjG2G:24-64,G:162-265
Q6XEC0n/a2RG6zrje6zrjH1H:24-64,H:162-265
Q6XEC0n/a2RG6zrje6zrjH2H:63-163