2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide
Q8N5Y8 — Protein mono-ADP-ribosyltransferase PARP16
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand UHB
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand UHB
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q8N5Y8 | n/a | 6hxr | UHB | A | 301 | e6hxrA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q8N5Y8 | n/a | 6hxr | UHB | A | 301 | e6hxrA2 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | ARTD15_N |
| Q8N5Y8 | n/a | 6hxr | UHB | B | 301 | e6hxrB1 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | ARTD15_N |
| Q8N5Y8 | n/a | 6hxr | UHB | B | 301 | e6hxrB2 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |