7-{5-[(3-{[(4-tert-butylphenyl)carbamoyl]amino}propyl)(propan-2-yl)amino]-5-deoxy-beta-D-ribofuranosyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Q8TEK3 — Histone-lysine N-methyltransferase, H3 lysine-79 specific
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 0QK
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 0QK
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q8TEK3 | n/a | 4eki | 0QK | A | 501 | e4ekiA1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 4er3 | 0QK | A | 401 | e4er3A1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 4er5 | 0QK | A | 502 | e4er5A1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |