N~6~-(2,6-dichlorophenyl)-N~6~-(pent-2-yn-1-yl)quinoline-4,6-diamine
Q8TEK3 — Histone-lysine N-methyltransferase, H3 lysine-79 specific
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 5JJ
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 5JJ
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q8TEK3 | n/a | 5mvs | 5JJ | A | 402 | e5mvsA1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 5mvs | 5JJ | B | 402 | e5mvsB1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 5mw3 | 5JJ | A | 401 | e5mw3A1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 5mw3 | 5JJ | B | 401 | e5mw3B1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |