~{N}1-[(~{S})-(3-chlorophenyl)-pyridin-2-yl-methyl]-4-methylsulfonyl-~{N}2-pyrimidin-2-yl-benzene-1,2-diamine
Q8TEK3 — Histone-lysine N-methyltransferase, H3 lysine-79 specific
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand N4W
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand N4W
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q8TEK3 | n/a | 6te6 | N4W | A | 401 | e6te6A1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6te6 | N4W | A | 401 | e6te6B1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6te6 | N4W | B | 401 | e6te6A1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6te6 | N4W | B | 401 | e6te6B1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |