3-[(4-azanyl-6-methoxy-1,3,5-triazin-2-yl)amino]-4-[[(~{S})-[2,2-bis(fluoranyl)-1,3-benzodioxol-4-yl]-(3-chloranylpyridin-2-yl)methyl]amino]benzenesulfonamide
Q8TEK3 — Histone-lysine N-methyltransferase, H3 lysine-79 specific
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand N5K
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand N5K
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q8TEK3 | n/a | 6ten | N5K | A | 401 | e6tenA1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6ten | N5K | A | 401 | e6tenB1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6ten | N5K | B | 401 | e6tenA1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |
| Q8TEK3 | n/a | 6ten | N5K | B | 401 | e6tenB1 | Rossmann-like | Rossmann-related | S-adenosyl-L-methionine-dependent methyltransferases | DOT1 |