8-(6-methoxypyridin-3-yl)-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]-5H-[1,2,3]triazolo[4,5-c]quinolin-4-one
Q9BVS4 — Serine/threonine-protein kinase RIO2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand 5ZH
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand 5ZH
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9BVS4 | n/a | 7vbt | 5ZH | A | 401 | e7vbtA1 | Protein kinase/SAICAR synthase/ATP-grasp | Protein kinase/SAICAR synthase/ATP-grasp | Protein kinase | RIO1 |
| Q9BVS4 | n/a | 7vbt | 5ZH | A | 401 | e7vbtA2 | HTH | HTH | winged helix domain | Rio2_N |
| Q9BVS4 | n/a | 7vbt | 5ZH | B | 401 | e7vbtB2 | Protein kinase/SAICAR synthase/ATP-grasp | Protein kinase/SAICAR synthase/ATP-grasp | Protein kinase | RIO1 |