~{N}-[3-[5-(5-ethoxypyridin-2-yl)-4-(2-fluorophenyl)-1,2,4-triazol-3-yl]cyclobutyl]pyridine-2-carboxamide
Q9H2K2 — Poly polymerase tankyrase-2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand N8K
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand N8K
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9H2K2 | n/a | 6tg4 | N8K | AAA | 1201 | e6tg4AAA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 6tg4 | N8K | BBB | 1201 | e6tg4BBB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 7pox | N8K | AAA | 1201 | e7poxAAA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 7pox | N8K | BBB | 1201 | e7poxBBB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |