~{N}-(2-methoxyphenyl)-4-[[2-(4-oxidanylidene-3~{H}-quinazolin-2-yl)ethyl-(thiophen-2-ylmethyl)carbamoyl]amino]benzamide
Q9H2K2 — Poly polymerase tankyrase-2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand OY6
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand OY6
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9H2K2 | n/a | 8b6m | OY6 | A | 1201 | e8b6mA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 8b6m | OY6 | A | 1201 | e8b6mB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 8b6m | OY6 | C | 1202 | e8b6mC1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 8b6m | OY6 | C | 1202 | e8b6mD1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | NADase_NGA |