2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide
Q9H2K2 — Poly polymerase tankyrase-2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand UHB
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand UHB
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9H2K2 | n/a | 4bj9 | UHB | A | 2165 | e4bj9A1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 4bj9 | UHB | B | 2165 | e4bj9B1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 4tk5 | UHB | A | 1202 | e4tk5A1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 4tk5 | UHB | B | 1202 | e4tk5B1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 4tk5 | UHB | C | 1202 | e4tk5C1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9H2K2 | n/a | 4tk5 | UHB | D | 1201 | e4tk5D1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |