(8S,9R)-5-fluoro-8-(4-fluorophenyl)-9-(1-methyl-1H-1,2,4-triazol-5-yl)-2,7,8,9-tetrahydro-3H-pyrido[4,3,2-de]phthalazin-3-one
Q9UGN5 — Poly polymerase 2 ADP-ribosyltransferase 2
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand DB11760
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand DB11760
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9UGN5 | DB11760 | 4pjv | 2YQ | A | 601 | e4pjvA1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9UGN5 | DB11760 | 4pjv | 2YQ | A | 601 | e4pjvA2 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | PARP_reg |
| Q9UGN5 | DB11760 | 4pjv | 2YQ | B | 601 | e4pjvB1 | ADP-ribosylation | ADP-ribosylation | ADP-ribosylation | PARP |
| Q9UGN5 | DB11760 | 4pjv | 2YQ | B | 601 | e4pjvB2 | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | Domain of poly(ADP-ribose) polymerase | PARP_reg |