(10R)-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]quinoline
Q9Y233 — cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand IV8
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand IV8
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9Y233 | n/a | 5sg1 | IV8 | A | 803 | e5sg1A1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sg1 | IV8 | B | 803 | e5sg1B1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sg1 | IV8 | C | 803 | e5sg1C1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sg1 | IV8 | D | 803 | e5sg1D1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |