N~4~-ethyl-5-[3-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine
Q9Y233 — cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand K3O
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand K3O
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9Y233 | n/a | 5sjj | K3O | A | 804 | e5sjjA1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjj | K3O | B | 803 | e5sjjB1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjj | K3O | C | 803 | e5sjjC1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjj | K3O | D | 803 | e5sjjD1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |