6-cyclopropyl-N-{(4S)-4-[(piperidin-1-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl}-3-[(pyrimidin-5-yl)amino]pyrazine-2-carboxamide
Q9Y233 — cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand K4U
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand K4U
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9Y233 | n/a | 5sju | K4U | A | 803 | e5sjuA1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sju | K4U | B | 803 | e5sjuB1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sju | K4U | C | 803 | e5sjuC1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sju | K4U | D | 803 | e5sjuD1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |