ethyl [(4-{[4-(azetidine-1-carbonyl)-1-methyl-1H-pyrazole-5-carbonyl]amino}-6-methylpyridin-2-yl)carbamothioyl]carbamate
Q9Y233 — cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand K6O
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand K6O
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9Y233 | n/a | 5sjp | K6O | A | 803 | e5sjpA1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjp | K6O | B | 803 | e5sjpB1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjp | K6O | C | 803 | e5sjpC1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5sjp | K6O | D | 803 | e5sjpD1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |