N-{[(4R)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-3-phenyl-1H-1,2,4-triazol-5-amine
Q9Y233 — cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
ECOD Domain Annotations
ECOD domains from AlphaFold model interacting with ligand KFX
| UniProt | DrugBank | PDB Ligand | Domain Label | ECOD ID | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|
| No predicted ECOD data found | ||||||||
ECOD domains from experimental PDB structures interacting with ligand KFX
| UniProt | DrugBank | PDB ID | Ligand Acc. | Chain | Res No. | Exp. Domain | X Group | H Group | T Group | F Group |
|---|---|---|---|---|---|---|---|---|---|---|
| Q9Y233 | n/a | 5ski | KFX | A | 803 | e5skiA1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5ski | KFX | B | 803 | e5skiB1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5ski | KFX | C | 803 | e5skiC1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |
| Q9Y233 | n/a | 5ski | KFX | D | 803 | e5skiD1 | PDEase-like | HD-domain/PDEase-like | HD-domain/PDEase-like | PDEase_I |