DB00734
Proteins interacting with this molecule.
| DrugDomain Data | DrugBank | PDB Ligand | UniProt | Protein Name | Drug Action | Affinity |
|---|---|---|---|---|---|---|
| Explore | DB00734 | 8NU | P08908 | 5-hydroxytryptamine receptor 1A | antagonist | Ki 21 nM | EC50 10000 nM |
| Explore | DB00734 | 8NU | P14416 | D dopamine receptor | antagonist | Ki 0.3 nM | IC50 3.6 nM |
| Explore | DB00734 | 8NU | P18089 | Alpha-2B adrenergic receptor | antagonist | Ki 8.5 nM |
| Explore | DB00734 | 8NU | P18825 | Alpha-2C adrenergic receptor | antagonist | Ki 1.3 nM |
| Explore | DB00734 | 8NU | P21728 | D dopamine receptor | antagonist | Ki 21 nM |
| Explore | DB00734 | 8NU | P28221 | 5-hydroxytryptamine receptor 1D | antagonist | Ki 3.9 nM |
| Explore | DB00734 | 8NU | P28223 | 5-hydroxytryptamine receptor 2A | antagonist | Ki 0.14 nM | IC50 0.707946 nM |
| Explore | DB00734 | 8NU | P28335 | 5-hydroxytryptamine receptor 2C | antagonist | Ki 2.4 nM | IC50 1.8 nM |
| Explore | DB00734 | 8NU | P34969 | 5-hydroxytryptamine receptor 7 | antagonist | Ki 0.4 nM |
| Explore | DB00734 | 8NU | P35348 | Alpha-1A adrenergic receptor | antagonist | Ki 0.7 nM | IC50 10 nM |
| Explore | DB00734 | 8NU | P35367 | Histamine H1 receptor | antagonist | Ki 2.6 nM | IC50 454 nM |
| Explore | DB00734 | 8NU | P35368 | Alpha-1B adrenergic receptor | antagonist | n/a |
Showing 12 of 12 interactions